• v
  • t
  • e
Adrenergic receptor modulators
α1
Agonists
  • 6-FNE
  • Amidephrine
  • Buspirone
  • Cirazoline
  • Corbadrine
  • Deoxyepinephrine (epinine, N-methyldopamine)
  • Desglymidodrine
  • Dexisometheptene
  • Dipivefrine
  • Dopamine
  • Droxidopa (L-DOPS)
  • Epinephrine
  • Etilefrine
  • Etilevodopa
  • Ethylnorepinephrine
  • Ibopamine
  • Indanidine
  • Isometheptene
  • L-DOPA (levodopa)
  • L-Phenylalanine
  • L-Tyrosine
  • Melevodopa
  • Metaraminol
  • Methoxamine
  • Methyldopa
  • Midodrine
  • Naphazoline
  • Norepinephrine
  • Octopamine
  • Oxymetazoline
  • Phenylephrine
  • Phenylpropanolamine
  • Synephrine
  • Tetryzoline
  • Tiamenidine
  • XP21279
  • Xylometazoline
Antagonists
  • Abanoquil
  • Ajmalicine
  • Alfuzosin
  • Anisodamine
  • Anisodine
  • Atiprosin
  • Atypical antipsychotics (e.g., brexpiprazole, clozapine, olanzapine, quetiapine, risperidone)
  • Benoxathian
  • Beta blockers (e.g., adimolol, amosulalol, arotinolol, carvedilol, eugenodilol, labetalol)
  • Buflomedil
  • Bunazosin
  • Corynanthine
  • Dapiprazole
  • Domesticine
  • Doxazosin
  • Ergolines (e.g., acetergamine, ergotamine, dihydroergotamine, lisuride, nicergoline, terguride)
  • Etoperidone
  • Fenspiride
  • Hydroxyzine
  • Indoramin
  • Ketanserin
  • L-765,314
  • mCPP
  • Mepiprazole
  • Metazosin
  • Monatepil
  • Moxisylyte
  • Naftopidil
  • Nantenine
  • Neldazosin
  • Niaprazine
  • Niguldipine
  • Pardoprunox
  • Pelanserin
  • Perlapine
  • Phendioxan
  • Phenoxybenzamine
  • Phentolamine
  • Phenylpiperazine antidepressants (e.g., hydroxynefazodone, nefazodone, trazodone, triazoledione)
  • Piperoxan
  • Prazosin
  • Quinazosin
  • Quinidine
  • Silodosin
  • Spegatrine
  • Spiperone
  • Talipexole
  • Tamsulosin
  • Terazosin
  • Tiodazosin
  • Tolazoline
  • Tetracyclic antidepressants (e.g., amoxapine, maprotiline, mianserin)
  • Tricyclic antidepressants (e.g., amitriptyline, clomipramine, doxepin, imipramine, trimipramine)
  • Trimazosin
  • Typical antipsychotics (e.g., chlorpromazine, fluphenazine, loxapine, thioridazine)
  • Urapidil
  • WB-4101
  • Zolertine
α2
Agonists
  • (R)-3-Nitrobiphenyline
  • 4-NEMD
  • 6-FNE
  • Amitraz
  • Apraclonidine
  • Brimonidine
  • Clonidine
  • Corbadrine
  • Deoxyepinephrine (epinine, N-methyldopamine)
  • Detomidine
  • Dexmedetomidine
  • Dihydroergotamine
  • Dipivefrine
  • Dopamine
  • Droxidopa (L-DOPS)
  • Etilevodopa
  • Ergotamine
  • Epinephrine
  • Etilefrine
  • Ethylnorepinephrine
  • Guanabenz
  • Guanfacine
  • Guanoxabenz
  • L-DOPA (levodopa)
  • L-Phenylalanine
  • L-Tyrosine
  • Ibopamine
  • Lofexidine
  • Medetomidine
  • Melevodopa
  • Methyldopa
  • Mivazerol
  • Moxonidine
  • Naphazoline
  • Norepinephrine
  • Oxymetazoline
  • Phenylpropanolamine
  • Piperoxan
  • PS75
  • Rezatomidine
  • Rilmenidine
  • Romifidine
  • Talipexole
  • Tasipimidine
  • Tetryzoline
  • Tiamenidine
  • Tizanidine
  • Tolonidine
  • Urapidil
  • Vatinoxan
  • XP21279
  • Xylazine
  • Xylometazoline
Antagonists
  • 1-PP
  • Adimolol
  • Amesergide
  • Aptazapine
  • Atipamezole
  • Atypical antipsychotics (e.g., asenapine, brexpiprazole, clozapine, lurasidone, olanzapine, paliperidone, quetiapine, risperidone, zotepine)
  • Azapirones (e.g., buspirone, gepirone, ipsapirone, tandospirone)
  • BRL-44408
  • Buflomedil
  • Cirazoline
  • Efaroxan
  • Esmirtazapine
  • Fenmetozole
  • Fluparoxan
  • Idazoxan
  • Ketanserin
  • Lisuride
  • mCPP
  • Mianserin
  • Mirtazapine
  • NAN-190
  • Pardoprunox
  • Phentolamine
  • Phenoxybenzamine
  • Piperoxan
  • Piribedil
  • Rauwolscine
  • Rotigotine
  • Setiptiline
  • Spegatrine
  • Spiroxatrine
  • Sunepitron
  • Terguride
  • Tolazoline
  • Typical antipsychotics (e.g., chlorpromazine, fluphenazine, loxapine, thioridazine)
  • Yohimbine
β
Agonists
  • Abediterol
  • Alifedrine
  • Amibegron
  • Arbutamine
  • Arformoterol
  • Arotinolol
  • BAAM
  • Bambuterol
  • Befunolol
  • Bitolterol
  • Broxaterol
  • Buphenine
  • Carbuterol
  • Carmoterol
  • Cimaterol
  • Clenbuterol
  • Colterol
  • Corbadrine
  • Denopamine
  • Deoxyepinephrine (epinine, N-methyldopamine)
  • Dipivefrine
  • Dobutamine
  • Dopamine
  • Dopexamine
  • Droxidopa (L-DOPS)
  • Epinephrine
  • Etafedrine
  • Etilefrine
  • Etilevodopa
  • Ethylnorepinephrine
  • Eugenodilol
  • Fenoterol
  • Formoterol
  • Hexoprenaline
  • Higenamine
  • Ibopamine
  • Indacaterol
  • Isoetarine
  • Isoprenaline
  • Isoxsuprine
  • L-DOPA (levodopa)
  • L-Phenylalanine
  • L-Tyrosine
  • Levosalbutamol
  • Lubabegron
  • Mabuterol
  • Melevodopa
  • Methoxyphenamine
  • Methyldopa
  • Mirabegron
  • Norepinephrine
  • Orciprenaline
  • Oxyfedrine
  • PF-610355
  • Phenylpropanolamine
  • Pirbuterol
  • Prenalterol
  • Ractopamine
  • Procaterol
  • Reproterol
  • Rimiterol
  • Ritodrine
  • Salbutamol
  • Salmeterol
  • Solabegron
  • Terbutaline
  • Tretoquinol
  • Tulobuterol
  • Vibegron
  • Vilanterol
  • Xamoterol
  • XP21279
  • Zilpaterol
  • Zinterol
Antagonists
  • Acebutolol
  • Adaprolol
  • Adimolol
  • Afurolol
  • Alprenolol
  • Alprenoxime
  • Amosulalol
  • Ancarolol
  • Arnolol
  • Arotinolol
  • Atenolol
  • Befunolol
  • Betaxolol
  • Bevantolol
  • Bisoprolol
  • Bopindolol
  • Bornaprolol
  • Brefonalol
  • Bucindolol
  • Bucumolol
  • Bufetolol
  • Bufuralol
  • Bunitrolol
  • Bunolol
  • Bupranolol
  • Butaxamine
  • Butidrine
  • Butofilolol
  • Capsinolol
  • Carazolol
  • Carpindolol
  • Carteolol
  • Carvedilol
  • Celiprolol
  • Cetamolol
  • Cicloprolol
  • Cinamolol
  • Cloranolol
  • Cyanopindolol
  • Dalbraminol
  • Dexpropranolol
  • Diacetolol
  • Dichloroisoprenaline
  • Dihydroalprenolol
  • Dilevalol
  • Diprafenone
  • Draquinolol
  • Ecastolol
  • Epanolol
  • Ericolol
  • Ersentilide
  • Esatenolol
  • Esprolol
  • Eugenodilol
  • Exaprolol
  • Falintolol
  • Flestolol
  • Flusoxolol
  • Hydroxycarteolol
  • Hydroxytertatolol
  • ICI-118,551
  • Idropranolol
  • Indenolol
  • Indopanolol
  • Iodocyanopindolol
  • Iprocrolol
  • Isoxaprolol
  • Isamoltane
  • Labetalol
  • Landiolol
  • Levobetaxolol
  • Levobunolol
  • Levomoprolol
  • Medroxalol
  • Mepindolol
  • Metipranolol
  • Metoprolol
  • Moprolol
  • Nadolol
  • Nadoxolol
  • Nebivolol
  • Nifenalol
  • Nipradilol
  • Oxprenolol
  • Pacrinolol
  • Pafenolol
  • Pamatolol
  • Pargolol
  • Penbutolol
  • Pindolol
  • Practolol
  • Primidolol
  • Procinolol
  • Pronethalol
  • Propafenone
  • Propranolol
  • Ridazolol
  • Ronactolol
  • Soquinolol
  • Sotalol
  • Spirendolol
  • SR 59230A
  • Sulfinalol
  • Talinolol
  • Tazolol
  • Tertatolol
  • Tienoxolol
  • Tilisolol
  • Timolol
  • Tiprenolol
  • Tolamolol
  • Toliprolol
  • Xibenolol
  • Xipranolol
  • See also: Receptor/signaling modulators
  • Dopaminergics
  • Serotonergics
  • Monoamine reuptake inhibitors
  • Monoamine releasing agents
  • Monoamine metabolism modulators
  • Monoamine neurotoxins
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